YEATS4 binder 4e

Chemical Structure : YEATS4 binder 4e

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货号: PC-49599Not For Human Use, Lab Use Only.

YEATS4 binder 4e is a potent, selective small-molecule epigenetic reader YEATS4 binder with Ki of 37 nM, >15-fold selectivity over YEATS1, 2 and 3.

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生物&药学活性

YEATS4 binder 4e is a potent, selective small-molecule epigenetic reader YEATS4 binder with Ki of 37 nM, >15-fold selectivity over YEATS1, 2 and 3.
YEATS4 binder 4e directly binds to YEATS4 at the lysine acetylation recognition site of the YEATS domain.
YEATS4 binder 4e engages YEATS4 with nanomolar potency in a whole-cell nanoluciferase bioluminescent resonance energy transfer assay (IC50=300 nM).

物理化学性质&存储条件

分子量	414.55
分子式	C23H34N4O3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-ethyl-3-((3R,4S)-1-((4-hydroxytetrahydro-2H-pyran-4-yl)methyl)-3-methylpiperidin-4-yl)-2-methylpyrazolo[1,5-a]pyridine-6-carboxamide

参考文献

1. Allyn T Londregan, et al. J Med Chem. 2022 Dec 23. doi: 10.1021/acs.jmedchem.2c01421.

YEATS4 binder 4e

生物&药学活性

物理化学性质&存储条件

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YEATS4 binder 4e

生物&药学活性

物理化学性质&存储条件

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