Y08284 | CBP/p300 inhibitor | Probechem Biochemicals

Chemical Structure : Y08284

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货号: PC-22485Not For Human Use, Lab Use Only.

Y08284 is a potent, selective CBP/p300 bromodomain inhibitor with IC50 of 4.21 nM (CBP bromodomain) in HTRF assays.

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Y08284 is a potent, selective CBP/p300 bromodomain inhibitor with IC50 of 4.21 nM (CBP bromodomain) in HTRF assays.

分子量	476.51
分子式	C26H25FN4O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
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Solubility	10 mM in DMSO
Chemical Name/SMILES	3-Acetyl-N-(3-(1-cyclopropyl-1H-pyrazol-4-yl)-2-fluoro-5-(1-hydroxyethyl)phenyl)-7-methoxyindolizine-1-carboxamide

1. Qiuping Xiang, et al. J Med Chem. 2022 Jan 13;65(1):785-810.