Azetukalner (XEN1101) | Kv7.2/Kv7.3 activator | Probechem Biochemicals

Chemical Structure : XEN1101

CAS No.: 1009344-33-5

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XEN1101 (Azetukalner, Encukalner)

货号: PC-73196Not For Human Use, Lab Use Only.

XEN1101 (Azetukalner) is a small molecule activator/opener of Kv7.2/Kv7.3 (KCNQ2/3) potassium channel with EC50 of 27 nM.

规格	价格	库存
10 mg	￥880	In stock
25 mg	￥1480	In stock
50 mg	￥2480	In stock
100 mg		Get quote

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生物&药学活性

XEN1101 (Azetukalner) is a small molecule activator/opener of Kv7.2/Kv7.3 (KCNQ2/3) potassium channel with EC50 of 27 nM.
XEN1101 (Azetukalner) is approximately 4-fold more selective for Kv7.2/7.3 over Kv7.3/7.5 (EC50 of 94 nM) and Kv7.4 (EC50 of 113 nM) channels.
XEN1101 (Azetukalner) also exhibits a selectivity >100-fold for Kv7 channels over other ion channels and receptors.

物理化学性质&存储条件

分子量	368.49
分子式	C23H29FN2O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(4-(6-Fluoro-3,4-dihydroisoquinolin-2(1H)-yl)-2,6-dimethylphenyl)-3,3-dimethylbutanamide

参考文献

1. Patent WO2021113757A1, compound A

XEN1101 (Azetukalner, Encukalner)

生物&药学活性

物理化学性质&存储条件

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XEN1101 (Azetukalner, Encukalner)

生物&药学活性

物理化学性质&存储条件

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