WIN 55,212-2 mesylate |CAS:131543-23-2 Probechem Biochemicals

Chemical Structure : WIN 55,212-2 mesylate

CAS No.: 131543-23-2

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WIN 55,212-2 mesylate ((R)-(+)-WIN 55212;WIN 55212-2)

货号: PC-43469Not For Human Use, Lab Use Only.

WIN 55,212-2 mesylate (WIN 55212-2) is a potent cannabinoid receptor agonist with Ki of 62.3 and 3.3 nM for human recombinant CB1 and CB2 receptors, respectively.

规格	价格	库存
25 mg	￥1280	In stock
50 mg	￥1980	In stock
100 mg	￥4580	In stock
500 mg		Get quote

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生物&药学活性

WIN 55,212-2 mesylate (WIN 55212-2) is a potent cannabinoid receptor agonist with Ki of 62.3 and 3.3 nM for human recombinant CB1 and CB2 receptors, respectively.
WIN 55,212-2 increases extracellular glutamate levels, displaying a bell-shaped concentration-response curve at 0.01-100 nM.
WIN 55,212-2 increases dialysate glutamate levels the prefrontal cortex from of the awake rats, also demonstrates anticonvulsant effect in vivo pre-treated with 20 mg/kg of pioglitazone.

物理化学性质&存储条件

分子量	522.61
分子式	C28H30N2O6S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
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Solubility	DMSO: ≥ 34 mg/mL
Chemical Name/SMILES	Methanone, [(3R)-2,3-dihydro-5-methyl-3-(4-morpholinylmethyl)pyrrolo[1,2,3-de]-1,4-benzoxazin-6-yl]-1-naphthalenyl-, methanesulfonate (1:1)

参考文献

1. Felder CC, et al. Mol Pharmacol. 1995 Sep;48(3):443-50.

2. Griffin G, et al. J Pharmacol Exp Ther. 1998 May;285(2):553-60.

3. D'Ambra TE, et al. J Med Chem. 1992 Jan;35(1):124-35.

4. Martellotta MC, et al. Neuroscience. 1998 Jul;85(2):327-30.

WIN 55,212-2 mesylate ((R)-(+)-WIN 55212;WIN 55212-2)

生物&药学活性

物理化学性质&存储条件

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WIN 55,212-2 mesylate ((R)-(+)-WIN 55212;WIN 55212-2)

生物&药学活性

物理化学性质&存储条件

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