欢迎访问ProbeChem中文网站，英文网站请访问www.probechem.com
    英文 |     中文

产品咨询: sales@probechem.com
订购: order@probechem.com

首页-小分子抑制剂&激动剂-GPCR-5-HT Receptor-VU6047534
VU6047534

Chemical Structure : VU6047534

CAS No.: 3029026-20-5

加入收藏

VU6047534 (VU 6047534)

货号: PC-21829Not For Human Use, Lab Use Only.

VU6047534 is a selective, peripherally restricted 5-HT2B partial agonist with IC50 of 480 nM in radioligand binding assays.

规格 价格 库存 数量
50 mg Get quote
100 mg Get quote
200 mg Get quote
获取报价单
* 请选择数量再加入购物车
 or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    VU6047534 is a selective, peripherally restricted 5-HT2B partial agonist with IC50 of 480 nM in radioligand binding assays.
    VU6047534 shows high subtype selectivity relative to 5-HT2A and 5-HT2C (no significant inhibition up to 10 uM).
    VU6047534 is peripherally restricted and able to both prevent and treat Sugen-hypoxia-induced pulmonary arterial hypertension.

    物理化学性质&存储条件

    分子量 351.42
    分子式 C19H17N3O2S
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20°C 12 个月; 4°C 6 个月
    配置液
    -80°C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    3-(1-methyl-1H-indol-5-yl)-5,6,7,8-tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione

    参考文献

    1. Valentine MS, et al. JACC Basic Transl Sci. 2023 Sep 13;8(10):1379-1388.

    备案号：沪ICP备16042516号-1 Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

    联系我们 sales@probechem.com

    Bulk Inquiry

    * Indicates a Required FieldYour information is safe with us.

    • *Product name:
    • *Applicant name:
    • *Email address:
    • *Organization name:
    • *Requested quantity:
    • *Country:
    • *Additional Information:

    询单

    • *产品名称:
    • *姓名:
    • *邮箱:
    • *公司名称:
    • *询单数量:
    • *国籍:
    • 询单信息: