VRK1 inhibitor Compound 1 (VRK1-IN-1)

Chemical Structure : VRK1 inhibitor Compound 1

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货号: PC-26316Not For Human Use, Lab Use Only.

VRK1 inhibitor Compound 1 (VRK1-IN-1) is a potent, selective and ATP-competitive inhibitor of Vaccinia-related kinase 1 (VRK1) with Ki of 82 nM and IC50 of 154 nM, selective for VRK1 over VRK2.

规格	价格	库存	数量
25 mg		Get quote
50 mg		Get quote
100 mg		Get quote

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生物&药学活性

VRK1 inhibitor Compound 1 (VRK1-IN-1) is a potent, selective and ATP-competitive inhibitor of Vaccinia-related kinase 1 (VRK1) with Ki of 82 nM and IC50 of 154 nM, selective for VRK1 over VRK2.

物理化学性质&存储条件

分子量	346.22
分子式	C14H13Cl2NO3S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(Z)-3-butyl-5-(3,5-dichloro-4-hydroxybenzylidene)thiazolidine-2,4-dione

参考文献

1. Crowley-Dolen EK, et al. J Biol Chem. 2026 Mar 6:111355.