VR23 | Proteasome inhibitor | Probechem Biochemicals

Chemical Structure : VR23

CAS No.: 1624602-30-7

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VR23 (Proteasome inhibitor VR23)

货号: PC-45547Not For Human Use, Lab Use Only.

VR23 is a potent inhibitor of trypsin-like proteasome (IC50=1 nM), chymotrypsin-like proteasome (IC50=50-100 nM) and caspase-like proteasome (IC50=3 uM).

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10 mg	￥880	In stock
25 mg	￥1380	In stock
50 mg	￥2280	In stock
100 mg	￥3780	In stock
250 mg		Get quote

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生物&药学活性

VR23 is a potent inhibitor of trypsin-like proteasome (IC50=1 nM), chymotrypsin-like proteasome (IC50=50-100 nM) and caspase-like proteasome (IC50=3 uM).
VR23 targets the β2 of the 20S proteasome catalytic subunit and structurally distinct from other known proteasome inhibitors and selectively kills cancer cells by apoptosis, with little effect on noncancerous cells.

物理化学性质&存储条件

分子量	477.8782
分子式	C19H16ClN5O6S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Quinoline, 7-chloro-4-[4-[(2,4-dinitrophenyl)sulfonyl]-1-piperazinyl]-

参考文献

1. Pundir S, et al. Cancer Res. 2015 Oct 1;75(19):4164-75.

VR23 (Proteasome inhibitor VR23)

生物&药学活性

物理化学性质&存储条件

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VR23 (Proteasome inhibitor VR23)

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物理化学性质&存储条件

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