VGSC blocker 1 |CAS: 2230472-55-4 Probechem Biochemicals

Chemical Structure : VGSC blocker 1

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VGSC blocker 1 (Nav1.5 inhibitor 1)

货号: PC-35117Not For Human Use, Lab Use Only.

VGSC blocker 1 is a potent, small molecule blocker of neonatal isoform of the VGSC subtype, Nav1.5 (nNav1.5), blocks INa peak currents 34.9% at 1 uM.

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25 mg		Get quote
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100 mg		Get quote

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生物&药学活性

VGSC blocker 1 is a potent, small molecule blocker of neonatal isoform of the VGSC subtype, Nav1.5 (nNav1.5), blocks INa peak currents 34.9% at 1 uM.
VGSC blocker 1 inhibits cell invasion 0.3% at 1 uM in human breast cancer cell line MDA-MB-231, without affecting the cell viability.

物理化学性质&存储条件

分子量	386.531
分子式	C24H32F2N2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	4,4-bis(4-fluorophenyl)-N-(3-(piperidin-1-yl)propyl)butan-1-amine

参考文献

1. Dutta S, et al. Bioorg Med Chem. 2018 May 15;26(9):2428-2436.

VGSC blocker 1 (Nav1.5 inhibitor 1)

生物&药学活性

物理化学性质&存储条件

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VGSC blocker 1 (Nav1.5 inhibitor 1)

生物&药学活性

物理化学性质&存储条件

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