UR-144 |CAS:1199943-44-6 Probechem Biochemicals

Chemical Structure : UR-144

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UR-144 (UR 144;UR144)

货号: PC-60762Not For Human Use, Lab Use Only.

UR-144 is a potent, selective full agonist of the peripheral cannabinoid receptor CB2 with Ki of 1.8 nM, >80-fold selectivity over CB1 (Ki=150 nM).

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生物&药学活性

UR-144 is a potent, selective full agonist of the peripheral cannabinoid receptor CB2 with Ki of 1.8 nM, >80-fold selectivity over CB1 (Ki=150 nM).
UR-144 possesses an EC50 of 421 nM for human CB1 receptors, and 72 nM for human CB2 receptors, produces bradycardia and hypothermia in rats at a dose of 10 mg/kg.

物理化学性质&存储条件

分子量	311.461
分子式	C21H29NO
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(1-Pentyl-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone

参考文献

1. Banister SD, et al. ACS Chem Neurosci. 2015 Aug 19;6(8):1445-58.

2. Dhopeshwarkar A, et al. J Pharmacol Exp Ther. 2016 Aug;358(2):342-51.

UR-144 (UR 144;UR144)

生物&药学活性

物理化学性质&存储条件

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UR-144 (UR 144;UR144)

生物&药学活性

物理化学性质&存储条件

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