UK-369003 (Gisadenafil besylate) | PDE5 inhibitor | Probechem Biochemicals

Chemical Structure : UK-369003

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UK-369003 (Gisadenafil besylate, UK369003)

货号: PC-61897Not For Human Use, Lab Use Only.

UK-369003 (Gisadenafil besylate) is a novel, potent, selective, orally bioavailable PDE5 inhibitor with IC50 of 1.23 nM, displays 117-fold selectivity over PDE6.

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生物&药学活性

UK-369003 (Gisadenafil besylate) is a novel, potent, selective, orally bioavailable PDE5 inhibitor with IC50 of 1.23 nM, displays 117-fold selectivity over PDE6.
UK-369003 demonstrates efficacy in patients with lower urinary tract symptoms (LUTS) associated with benign prostatic hyperplasia (BPH).

物理化学性质&存储条件

分子量	677.79
分子式	C23H33N7O5S.C6H6O3S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	5-[2-Ethoxy-5-[(4-ethyl-1-piperazinyl)sulfonyl]-3-pyridinyl]-3-ethyl-2,6-dihydro-2-(2-methoxyethyl)-7H-pyrazolo[4,3-d]pyrimidin-7-one benzenesulfonate

参考文献

1. Rawson DJ, et al. Bioorg Med Chem. 2012 Jan 1;20(1):498-509.

2. Martínez-Salamanca JI, et al. Eur Urol. 2011 Sep;60(3):527-35.

3. Watson KJ, et al. Drug Metab Dispos. 2011 Jul;39(7):1203-13.

UK-369003 (Gisadenafil besylate, UK369003)

生物&药学活性

物理化学性质&存储条件

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UK-369003 (Gisadenafil besylate, UK369003)

生物&药学活性

物理化学性质&存储条件

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