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首页-小分子抑制剂&激动剂-Membrane Transporter/Ion Channel-Glutamate Transporter-UCPH-102
UCPH-102

Chemical Structure : UCPH-102

CAS No.: 1229591-56-3

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UCPH-102 (UCPH102)

货号: PC-62149Not For Human Use, Lab Use Only.

UCPH-102 is a selective, brain penetrant inhibitor of EAAT1 (Excitatory amino acid transporter 1) with IC50 of 420 nM.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    UCPH-102 is a selective, brain penetrant inhibitor of EAAT1 (Excitatory amino acid transporter 1) with IC50 of 420 nM.
    UCPH-102 exhibits no inhibitory activity aganist EAAT2-5 (>300 uM).
    UCPH-102 has been shown to cross the blood-brain barrier, and become a valuable tool for studying the role of EAAT1 in brain.

    物理化学性质&存储条件

    分子量 330.387
    分子式 C21H18N2O2
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    2-Amino-5,6,7,8-tetrahydro-4-methyl-7-(1-naphthalenyl)-5-oxo-4H-1-benzopyran-3-carbonitrile

    参考文献

    1. Huynh TH, et al. Bioorg Med Chem. 2012 Dec 1;20(23):6831-9.

    2. Haym I, et al. ChemMedChem. 2016 Feb 17;11(4):403-19.

    3. Erichsen MN, et al. Neurochem Res. 2014 Oct;39(10):1964-79.

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