Tonapofylline |CAS:340021-17-2 Probechem Biochemicals

Chemical Structure : Tonapofylline

CAS No.: 340021-17-2

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Tonapofylline (BG 9928;BG9928)

货号: PC-60741Not For Human Use, Lab Use Only.

Tonapofylline (BG9928) is a potent, selective and orally bioavailable adenosine A1 (A1A) receptor antagonist with Ki of 7 nM.

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10 mg	￥2480	In stock
25 mg	￥4280	In stock
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生物&药学活性

Tonapofylline (BG9928) is a potent, selective and orally bioavailable adenosine A1 (A1A) receptor antagonist with Ki of 7 nM.
Tonapofylline (BG9928) displays 915-foldselectivity over A2A receptor, 12-fold over A2B receptor.
Tonapofylline (BG9928) increases sodium excretion and cause natriuresis without causing kaliuresis or reducing renal function.

物理化学性质&存储条件

分子量	416.522
分子式	C22H32N4O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1,3-dipropyl-8-[1-(4-propionate)-bicyclo-[2,2,2]octyl]xanthine

参考文献

1. Auchampach JA, et al. J Pharmacol Exp Ther. 2004 Mar;308(3):846-56.

2. Kiesman WF, et al. J Med Chem. 2006 Nov 30;49(24):7119-31.

3. Greenberg B, et al. J Am Coll Cardiol. 2007 Aug 14;50(7):600-6.

Tonapofylline (BG 9928;BG9928)

生物&药学活性

物理化学性质&存储条件

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Tonapofylline (BG 9928;BG9928)

生物&药学活性

物理化学性质&存储条件

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