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首页-小分子抑制剂&激动剂-Membrane Transporter/Ion Channel-GABA Transporter (GAT)-Tiagabine hydrochloride
Tiagabine hydrochloride

Chemical Structure : Tiagabine hydrochloride

CAS No.: 145821-59-6

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Tiagabine hydrochloride (NO050328, NO328)

货号: PC-24080Not For Human Use, Lab Use Only.

Tiagabine hydrochloride is an anticonvulsant agent and selective inhibitor of
GABA transporter 1 (GAT1) with Ki of 0.1 uM, potently and selectively inhibits GABA reuptake with IC50 of 67, 446 and 182 nM for [3H]GABA uptake in synaptosomes, neurons and glia, respectively.

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10 mg ￥480 In stock
50 mg ￥980 In stock
100 mg ￥1480 In stock
250 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Tiagabine hydrochloride is an anticonvulsant agent and selective inhibitor of
GABA transporter 1 (GAT1) with Ki of 0.1 uM, potently and selectively inhibits GABA reuptake with IC50 of 67, 446 and 182 nM for [3H]GABA uptake in synaptosomes, neurons and glia, respectively.

物理化学性质&存储条件

分子量 412.00
分子式 C20H26ClNO2S2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(R)-1-(4,4-Bis(3-methylthiophen-2-yl)but-3-en-1-yl)piperidine-3-carboxylic acid hydrochloride

参考文献

1. Braestrup C, et al. J Neurochem. 1990 Feb;54(2):639-47.

2. Henjum S, Neurochem Int. 2007 Jan;50(2):365-70.

3. Sheehan DV, et al. Psychopharmacol Bull. 2007;40(3):32-40.

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