Tenalisib |CAS:1639417-53-0 Probechem Biochemicals

Chemical Structure : Tenalisib

CAS No.: 1639417-53-0

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Tenalisib (RP-6530;RP 6530;RP6530)

货号: PC-60567Not For Human Use, Lab Use Only.

Tenalisib (RP-6530) is a potent, selective, orally active p110δ/γ PI3K dual inhibitor with IC50 of 24.5 and 33.2 nM, respectively.

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25 mg	￥2180	In stock
50 mg	￥3780	In stock
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生物&药学活性

Tenalisib (RP-6530) is a potent, selective, orally active p110δ/γ PI3K dual inhibitor with IC50 of 24.5 and 33.2 nM, respectively.
Tenalisib (RP-6530) displays good selectivity over p110α (>300-fold) and p110β (>100-fold) isoforms.
Tenalisib (RP-6530) inhibits LPS induced CD19+ cell proliferation in human whole blood with EC50 of 250 nM, and LPS induced CD45R+ cell proliferation in mouse whole blood with EC50 of 101 nM.
Tenalisib (RP-6530) shows the potential for treatment of cancer and inflammation diseases.

物理化学性质&存储条件

分子量	415.43
分子式	C23H18FN5O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-2-(1-((7H-purin-6-yl)amino)propyl)-3-(3-fluorophenyl)-4H-chromen-4-one

Tenalisib (RP-6530;RP 6530;RP6530)

生物&药学活性

物理化学性质&存储条件

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Tenalisib (RP-6530;RP 6530;RP6530)

生物&药学活性

物理化学性质&存储条件

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