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首页-小分子抑制剂&激动剂-Nuclear Receptor/Transcription Factor-Progesterone Receptor-Tanaproget
Tanaproget

Chemical Structure : Tanaproget

CAS No.: 304853-42-7

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Tanaproget (NSP-989, NSP989, WAY-166989, WAY166989)

货号: PC-27686Not For Human Use, Lab Use Only.

Tanaproget (NSP-989, WAY-166989) is a potent and selective, nonsteroidal progesterone receptor (PR) agonist with EC50 of 0.15 nM, displaces [3H]R5020 (synthetic steroidal progestin) binding to the human PR with IC50 of 1.7 nM.

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25 mg ￥1580 In stock
50 mg ￥2580 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Tanaproget (NSP-989, WAY-166989) is a potent and selective, nonsteroidal progesterone receptor (PR) agonist with EC50 of 0.15 nM, displaces [3H]R5020 (synthetic steroidal progestin) binding to the human PR with IC50 of 1.7 nM.
Tanaproget promotes PR and SRC-1 interaction in mammalian cells.
Tanaproget shows 0.3-0.5 nM affinity for monkey, rat, and rabbit PR.
Tanaproget does not exhibit any agonist activity against other steroid receptors ER, AR, and GR.

物理化学性质&存储条件

分子量 297.38
分子式 C16H15N3OS
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

5-(4,4-dimethyl-2-thioxo-1,4-dihydro-2H-benzo[d][1,3]oxazin-6-yl)-1-methyl-1H-pyrrole-2-carbonitrile

参考文献

1. Zhang Z, et al. J Biol Chem. 2005 Aug 5;280(31):28468-75.

2. Fensome A, et al. J Med Chem. 2005 Aug 11;48(16):5092-5.

3. Bapst JL, et al. Contraception. 2006 Nov;74(5):414-8.

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