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首页-小分子抑制剂&激动剂-GPCR-Free Fatty Acid Receptor (FFAR)-TUG-1958
TUG-1958

Chemical Structure : TUG-1958

CAS No.: 3032285-22-3

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TUG-1958 (TUG1958)

货号: PC-24798Not For Human Use, Lab Use Only.

TUG-1958 is a potent, selective antagonist of GPR43 (FFA2R, free fatty acid receptor 2) with pIC50 of 7.41 uM (hFFA2) in [35S]GTPγS-based binding assays.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

TUG-1958 is a potent, selective antagonist of GPR43 (FFA2R, free fatty acid receptor 2) with pIC50 of 7.41 uM (hFFA2) in [35S]GTPγS-based binding assays.
TUG-1958 is completely selective over the related receptor FFA3 with no sign of activity up to 100 μM.
TUG-1958 has excellent solubility and favorable pharmacokinetic properties.

物理化学性质&存储条件

分子量 397.37
分子式 C20H19F4NO3
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(R)-4-(2-(3-fluorophenyl)acetamido)-5-(4-(trifluoromethyl)phenyl)pentanoic acid

参考文献

1. Højgaard Hansen A, et al. ChemMedChem. 2021 Nov 5;16(21):3326-3341.

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