TP-238 | 2415263-04-4 Probechem Biochemicals

Chemical Structure : TP-238

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TP-238 (TP238)

货号: PC-35848Not For Human Use, Lab Use Only.

TP-238 (TP238) is a CECR2/BPTF bromodomains chemical probe with IC50 of 30 nM against CECR2 and 350 nM against BPTF in an alphascreen assay, KD of 10 nM for CECR2 and 120nM for BPTF in ITC assays.

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生物&药学活性

TP-238 (TP238) is a CECR2/BPTF bromodomains chemical probe with IC50 of 30nM against CECR2 and 350 nM against BPTF in an alphascreen assay, KD of 10 nM for CECR2 and 120 nM for BPTF in ITC assays.
TP-238 has been profiled against the panel of 338 kinases and showed no activity at 1 uM, the closest off-target bromodomain inhibition is BRD9 with IC50 of 1.4 uM.

物理化学性质&存储条件

分子量	458.581
分子式	C22H30N6O3S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(3-(1H-pyrazol-1-yl)propyl)-6-(4-(3-(dimethylamino)propoxy)phenyl)-2-(methylsulfonyl)pyrimidin-4-amine

TP-238 (TP238)

生物&药学活性

物理化学性质&存储条件

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TP-238 (TP238)

生物&药学活性

物理化学性质&存储条件

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