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首页-小分子抑制剂&激动剂-Nuclear Receptor/Transcription Factor-PPAR-TIPP-204
TIPP-204

Chemical Structure : TIPP-204

CAS No.: 943544-10-3

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TIPP-204 (TIPP204)

货号: PC-23874Not For Human Use, Lab Use Only.

TIPP-204 is a potent, selective PPARδ agonist with EC50 of 0.91 nM, >250-fold selective PPARα and PPARγ.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

TIPP-204 is a potent, selective PPARδ agonist with EC50 of 0.91 nM, >250-fold selective PPARα and PPARγ.
TIPP-204 exhibits extremely potent PPARδ transactivation activity, comparable with or somewhat superior to that of the known PPARδ-selective agonist GW-501516.
TIPP-204 does not significantly activate VDR, PPARγ, LXRα, RARα or RXRα at concentrations up to 300 nM.
TIPP-204 regulated the expression of genes involved in lipid and glucose homeostasis.

物理化学性质&存储条件

分子量 469.48
分子式 C24H27F4NO4
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(S)-2-(4-butoxy-3-((2-fluoro-4-(trifluoromethyl)benzamido)methyl)benzyl)butanoic acid

参考文献

1. Kasuga J, et al. Bioorg Med Chem. 2007 Aug 1;15(15):5177-90.

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