THIQ | MC4R agonist | Probechem Biochemicals

Chemical Structure : THIQ

CAS No.: 312637-48-2

加入收藏

THIQ (MC4R agonist THIQ)

货号: PC-70060Not For Human Use, Lab Use Only.

THIQ is a potent and selective melanocortin 4 receptor (MC4R) agonist with EC50 of 2.1 nM.

规格	价格	库存
5 mg	￥980	In stock
10 mg	￥1580	In stock
25 mg	￥2780	In stock
50 mg	￥4580	In stock
100 mg		Get quote

获取报价单

* 请选择数量再加入购物车

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

生物&药学活性

THIQ is a potent and selective melanocortin 4 receptor (MC4R) agonist with EC50 of 2.1 nM.
THIQ has high selectivity over other melanocortin receptors (1184-fold vs MC3R, 350-fold vs MC5R).
THIQ enhances intracavernosal pressure and stimulates erectile activity in rats ex copula.

物理化学性质&存储条件

分子量	589.181
分子式	C33H41ClN6O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-N-((R)-1-(4-((1H-1,2,4-triazol-1-yl)methyl)-4-cyclohexylpiperidin-1-yl)-3-(4-chlorophenyl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide

参考文献

1. Sebhat IK, et al. J Med Chem. 2002 Oct 10;45(21):4589-93.

2. Martin WJ, et al. Eur J Pharmacol. 2002 Nov 1;454(1):71-9.

3. Molden BM, et al. Mol Endocrinol. 2015 Nov;29(11):1619-33.

THIQ (MC4R agonist THIQ)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

THIQ (MC4R agonist THIQ)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Get Quotation Now

* Indicates a Required FieldYour information is safe with us.