TGR-1202 R-enantiomer |CAS:1532533-69-9 Probechem Biochemicals

Chemical Structure : TGR-1202 R-enantiomer

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TGR-1202 R-enantiomer (RP5264 R-enantiomer;TGR1202 R-enantiomer)

货号: PC-42943Not For Human Use, Lab Use Only.

TGR-1202 R-enantiomer is is the less active enantiomer of TGR-1202 (Umbralisib), TGR-1202 is a potent, selective, orally available PI3Kδ inhibitor with IC50 of 22 nM..

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生物&药学活性

TGR-1202 R-enantiomer is is the less active enantiomer of TGR-1202 (Umbralisib), TGR-1202 is a potent, selective, orally available PI3Kδ inhibitor with IC50 of 22 nM.

物理化学性质&存储条件

分子量	571.5492
分子式	C31H24F3N5O3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	4H-1-Benzopyran-4-one, 2-[(1R)-1-[4-amino-3-[3-fluoro-4-(1-methylethoxy)phenyl]-1H-pyrazolo[3,4-d]pyrimidin-1-yl]ethyl]-6-fluoro-3-(3-fluorophenyl)-

参考文献

1. Locatelli SL, et al. Leukemia. 2016 Dec;30(12):2402-2405.

2. Deng C, et al. Blood. 2017 Jan 5;129(1):88-99.

3. Burris HA 3rd, et al. Lancet Oncol. 2018 Feb 20. pii: S1470-2045(18)30082-2.

4. Lampson BL, et al. Expert Opin Investig Drugs. 2017 Nov;26(11):1267-1279.

TGR-1202 R-enantiomer (RP5264 R-enantiomer;TGR1202 R-enantiomer)

生物&药学活性

物理化学性质&存储条件

参考文献

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TGR-1202 R-enantiomer (RP5264 R-enantiomer;TGR1202 R-enantiomer)

生物&药学活性

物理化学性质&存储条件

参考文献

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