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首页-小分子抑制剂&激动剂-GPCR-Prostaglandin Receptor-TG4-155
TG4-155

Chemical Structure : TG4-155

CAS No.: 1164462-05-8

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TG4-155 (TG 4-155)

货号: PC-62029Not For Human Use, Lab Use Only.

TG4-155 is a potent and selective prostaglandin EP2 receptor antagonist with Kb of 2.4 nM.

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10 mg ￥1280 In stock
25 mg ￥2180 In stock
50 mg ￥3580 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

TG4-155 is a potent and selective prostaglandin EP2 receptor antagonist with Kb of 2.4 nM.
TG4-155 displays 4,730-fold selectivity over EP4, >500-fold selectivity over human BLT1, EP1, EP3, and FP receptors, and 7-fold selectivity against human DP1 receptor.
TG4-155 displays robust inhibition of PGE2-induced cAMP accumulation in C6G cells stably expressing mouse EP2 receptor.
TG4-155 significantly reduces SE-induced neurodegeneration in mice.

物理化学性质&存储条件

分子量 394.5
分子式 C23H26N2O4
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(2E)-N-[2-(2-methyl-1H-indol-1-yl)ethyl]-3-(3,4,5-trimethoxyphenyl)-2-propenamide

参考文献

1. Jiang J, et al. Proc Natl Acad Sci U S A. 2012 Feb 21;109(8):3149-54.

2. Jiang J, et al. J Pharmacol Exp Ther. 2013 Feb;344(2):360-7.

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