TCS-OX2-29 | OX2R antagonist | Probechem Biochemicals

Chemical Structure : TCS-OX2-29

CAS No.: 372523-75-6

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TCS-OX2-29 (TCS OX2 29)

货号: PC-42159Not For Human Use, Lab Use Only.

TCS-OX2-29 is a potent, selective orexin-2 receptor (OX2R) antagonist with IC50 of 40 nM.

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10 mg	￥980	In stock
25 mg	￥1580	In stock
50 mg	￥2580	In stock
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生物&药学活性

TCS-OX2-29 is a potent, selective orexin-2 receptor (OX2R) antagonist with IC50 of 40 nM.
TCS-OX2-29 displays >250-fold selectivity for OX2 over OX1 and a panel of receptors, ion channels and transporters.
TCS-OX2-29 blocks the inhibitory action of orexin A on forskolin-induced cAMP formation.

物理化学性质&存储条件

分子量	397.5105
分子式	C23H31N3O3
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1-Butanone, 1-(3,4-dihydro-6,7-dimethoxy-2(1H)-isoquinolinyl)-3,3-dimethyl-2-[(4-pyridinylmethyl)amino]-, (2S)-

参考文献

1. Hirose M, et al. Bioorg Med Chem Lett. 2003 Dec 15;13(24):4497-9.

2. Urbańska A, et al. J Mol Neurosci. 2012 Jan;46(1):10-7.

3. Huang SC, et al. J Pharmacol Exp Ther. 2010 Aug;334(2):522-9.

TCS-OX2-29 (TCS OX2 29)

生物&药学活性

物理化学性质&存储条件

参考文献

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TCS-OX2-29 (TCS OX2 29)

生物&药学活性

物理化学性质&存储条件

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