TAK-802 hydrochloride | AChE inhibitor | Probechem Biochemicals

Chemical Structure : TAK-802 hydrochloride

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TAK-802 hydrochloride (TAK 802, TAK802)

货号: PC-61036Not For Human Use, Lab Use Only.

TAK-802 hydrochloride is a potent acetylcholinesterase (AChE) inhibitor with IC50 of 1.3 nM.

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25 mg		Get quote
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100 mg		Get quote

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生物&药学活性

TAK-802 hydrochloride is a potent acetylcholinesterase (AChE) inhibitor with IC50 of 1.3 nM.
TAK-802 exhibits high selectivity for acetylcholinesterase inhibition over butyrylcholinesterase inhibition.
TAK-802 increases rhythmic bladder contractions in Guinea pigs and rats without affecting the basal intravesical pressure.

物理化学性质&存储条件

分子量	456.986
分子式	C26H30ClFN2O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	8-[3-[1-[(3-fluorophenyl)methyl]-4-piperidinyl]-1-oxopropyl]-1,2,5,6-tetrahydro-4H-pyrrolo[3,2,1-ij]quinolin-4-one hydrochloride

参考文献

1. Ishichi Y, et al. Bioorg Med Chem. 2005 Mar 15;13(6):1901-11.

2. Nagabukuro H, et al. Eur J Pharmacol. 2004 Feb 6;485(1-3):299-305.

3. Nagabukuro H, et al. Eur J Pharmacol. 2004 Jun 28;494(2-3):225-32.

TAK-802 hydrochloride (TAK 802, TAK802)

生物&药学活性

物理化学性质&存储条件

参考文献

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TAK-802 hydrochloride (TAK 802, TAK802)

生物&药学活性

物理化学性质&存储条件

参考文献

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