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首页-小分子抑制剂&激动剂-Membrane Transporter/Ion Channel-GABA Receptor-Stiripentol
Stiripentol

Chemical Structure : Stiripentol

CAS No.: 49763-96-4

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Stiripentol (BCX2600, BCX-2600)

货号: PC-28175Not For Human Use, Lab Use Only.

Stiripentol (BCX2600) is an antiepileptic drug that acts directly on GABA(A) receptor as a positive allosteric modulator, also is an lactate dehydrogenase (LDH) inhibitor, inhibits lactate production and decreases glioblastoma invasion and growth.

规格 价格 库存 数量
25 mg ￥980 In stock
50 mg ￥1480 In stock
100 mg ￥2480 In stock
250 mg ￥3980 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Stiripentol (BCX2600) is an antiepileptic drug that acts directly on GABA(A) receptor as a positive allosteric modulator, also is an lactate dehydrogenase (LDH) inhibitor, inhibits lactate production and decreases glioblastoma invasion and growth.
Stiripentol can cross the blood–brain barrier for inhibiting cerebral LDHA/B activity in preclinical therapy studies in mice.
Stiripentol (150 mg/kg, i.p.) significantly increased survival in P3 tumor‐bearing mice.
Stiripentol induced genetic and metabolic alterations in GBM cells.
Stiripentol strongly suppressed drug-resistant epilepsy in animal model.

物理化学性质&存储条件

分子量 234.30
分子式 C14H18O3
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

1-(Benzo[d][1,3]dioxol-5-yl)-4,4-dimethylpent-1-en-3-ol

参考文献

1. Sada N, et al. Science. 2015 Mar 20;347(6228):1362-7.

2. Fisher JL. Neuropharmacology. 2009 Jan;56(1):190-7.

3. Guyon J, et al. EMBO Mol Med. 2022 Dec 7;14(12):e15343.

4. Yadav A, et al. Eur J Pharmacol. 2026 May 15;1024:178893.

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