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首页-小分子抑制剂&激动剂-JAK/STAT Signaling-JAK-Solcitinib
Solcitinib

Chemical Structure : Solcitinib

CAS No.: 1206163-45-2

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Solcitinib (GSK-2586184, GLPG-0778, GSK2586184, GLPG0778)

货号: PC-45072Not For Human Use, Lab Use Only.

Solcitinib (GSK2586184, GLPG0778) is a potent, selective and orally active JAK1 inhibitor with IC50 of 9.8 nM.

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5 mg (Free Sample) ￥280 In stock
25 mg ￥1580 In stock
50 mg ￥2380 In stock
100 mg ￥3880 In stock
250 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Solcitinib (GSK2586184, GLPG0778) is a potent, selective and orally active JAK1 inhibitor with IC50 of 9.8 nM.
Solcitinib (GSK2586184, GLPG0778) displays 11-, 55- and 23-fold selectivity over JAK2, JAK3 and TYK2, respectively.
Solcitinib (GSK2586184, GLPG0778) shows potential for the treatment of psoriasis, lupus, and ulcerative colitis.

物理化学性质&存储条件

分子量 389.4503
分子式 C22H23N5O2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

DMSO: 20 mg/mL
Chemical Name/SMILES

Cyclopropanecarboxamide, N-[5-[4-[(3,3-dimethyl-1-azetidinyl)carbonyl]phenyl][1,2,4]triazolo[1,5-a]pyridin-2-yl]-

参考文献

1. Ludbrook VJ, et al. Br J Dermatol. 2016 May;174(5):985-95. 

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