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首页-小分子抑制剂&激动剂-Metabolic Enzyme/Protease-Factor Xa-Segatroxaban
Segatroxaban

Chemical Structure : Segatroxaban

CAS No.: 1184300-63-7

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Segatroxaban (SAR107375E)

货号: PC-24866Not For Human Use, Lab Use Only.

Segatroxaban (SAR107375E) is a potent and highly selective dual FIIa/Xa inhibitor with Ki values of 8 nM and 1 nM on FIIa and FXa, IC50 values of 0.3/0.7 nM (FIIa/FXa) in buffer and of 16/3 nM (FIIa/FXa) in plasma, respectively.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

Segatroxaban (SAR107375E) is a potent and highly selective dual FIIa/Xa inhibitor with Ki values of 8 nM and 1 nM on FIIa and FXa, IC50 values of 0.3/0.7 nM (FIIa/FXa) in buffer and of 16/3 nM (FIIa/FXa) in plasma, respectively.

物理化学性质&存储条件

分子量 568.10
分子式 C24H30ClN5O5S2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2-Thiophenecarboxamide, 5-chloro-N-[(2S)-2-[[[2-methyl-3-(2-oxo-1-pyrrolidinyl)phenyl]sulfonyl]amino]-3-(4-methyl-1-piperazinyl)-3-oxopropyl]-

参考文献

1. Beck H, et al. J Med Chem. 2025 Jun 11. doi: 10.1021/acs.jmedchem.5c00538.

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