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首页-小分子抑制剂&激动剂-Metabolic Enzyme/Protease-Dipeptidyl Peptidase (DPP)-Saxagliptin
Saxagliptin

Chemical Structure : Saxagliptin

CAS No.: 361442-04-8

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Saxagliptin (BMS-477118;BMS 477118;BMS477118)

货号: PC-42509Not For Human Use, Lab Use Only.

Saxagliptin (BMS-477118) is a highly potent, long-acting, orally active DPP4 inhibitor with Ki of 0.6 nM.

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25 mg ￥780 In stock
50 mg ￥1180 In stock
100 mg ￥1980 In stock
250 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Saxagliptin (BMS-477118) is a highly potent, long-acting, orally active DPP4 inhibitor with Ki of 0.6 nM.
Saxagliptin (BMS-477118) shows no CYP3A4 inhibition up to 100 uM, and good oral exposure.

物理化学性质&存储条件

分子量 315.41
分子式 C18H25N3O2
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

DMSO: ≥ 34 mg/mL
Chemical Name/SMILES

2-Azabicyclo[3.1.0]hexane-3-carbonitrile, 2-[(2S)-2-amino-2-(3-hydroxytricyclo[3.3.1.13,7]dec-1-yl)acetyl]-, (1S,3S,5S)-

参考文献

1. Augeri DJ, et al. J Med Chem. 2005 Jul 28;48(15):5025-37.

2. Kim YB, et al. Arch Biochem Biophys. 2006 Jan 1;445(1):9-18.

3. Ikeda J, et al. J Pharmacol Sci. 2016 Sep;132(1):65-70.

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