SUCNR1 inhibitor 20 | SUCNR1 (GPR91) antagonist | Probechem Biochemicals

Chemical Structure : SUCNR1 inhibitor 20

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SUCNR1 inhibitor 20 (GPR91 antagonist)

货号: PC-72380Not For Human Use, Lab Use Only.

SUCNR1 inhibitor 20 is a potent, selective inhibitor (antagonist) of GPCR SUCNR1 (succinate receptor 1/GPR91) with IC50 of 88 nM.

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生物&药学活性

SUCNR1 inhibitor 20 is a potent, selective inhibitor (antagonist) of GPCR SUCNR1 (succinate receptor 1/GPR91) with IC50 of 88 nM.
SUCNR1 (GPR91) senses the citric cycle intermediate succinate and is implicated in various pathological conditions such as rheumatoid arthritis, liver fibrosis, or obesity.

物理化学性质&存储条件

分子量	518.917
分子式	C26H22ClF3N2O4
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-2-(2-(4'-chloro-2,2'-difluoro-5'-(piperidin-3-yloxy)-[1,1'-biphenyl]-3-carboxamido)-5-fluorophenyl)acetic acid

参考文献

1. Juraj Velcicky, et al. J Med Chem. 2020 Sep 10;63(17):9856-9875.

SUCNR1 inhibitor 20 (GPR91 antagonist)

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物理化学性质&存储条件

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SUCNR1 inhibitor 20 (GPR91 antagonist)

生物&药学活性

物理化学性质&存储条件

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