欢迎访问ProbeChem中文网站，英文网站请访问www.probechem.com
    英文 |     中文

产品咨询: sales@probechem.com
订购: order@probechem.com

首页-小分子抑制剂&激动剂-Metabolic Enzyme/Protease-Steroid Sulfatase (STS)-STX681
STX681

Chemical Structure : STX681

CAS No.: 537674-89-8

加入收藏

STX681 (STX-681)

货号: PC-61432Not For Human Use, Lab Use Only.

STX681 is a potent, orally active, dual-acting aromatase and steroid sulfatase (STS) inhibitor with IC50 of 0.82 nM and 39 nM, respectively.

规格 价格 库存 数量
25 mg Get quote
50 mg Get quote
100 mg Get quote
获取报价单
* 请选择数量再加入购物车
 or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    STX681 is a potent, orally active, dual-acting aromatase and steroid sulfatase (STS) inhibitor with IC50 of 0.82 nM and 39 nM, respectively.
    STX681 significantly reduces plasma E2 levels, completely inhibits the growth of both MCF-7(STS) tumor growth and MCF-7(AROM) tumor in a xenograft nude mouse model.

    物理化学性质&存储条件

    分子量 449.283
    分子式 C16H13BrN6O3S
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    Sulfamic acid, 2-bromo-4-[[(4-cyanophenyl)-4H-1,2,4-triazol-4-ylamino]methyl]phenyl ester

    参考文献

    1. Foster PA, et al. Clin Cancer Res. 2008 Oct 15;14(20):6469-77.

    2. Woo LW, et al. J Med Chem. 2007 Jul 26;50(15):3540-60.

    备案号：沪ICP备16042516号-1 Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

    联系我们 sales@probechem.com

    Bulk Inquiry

    * Indicates a Required FieldYour information is safe with us.

    • *Product name:
    • *Applicant name:
    • *Email address:
    • *Organization name:
    • *Requested quantity:
    • *Country:
    • *Additional Information:

    询单

    • *产品名称:
    • *姓名:
    • *邮箱:
    • *公司名称:
    • *询单数量:
    • *国籍:
    • 询单信息: