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首页-小分子抑制剂&激动剂-GPCR-Opioid Receptor-SR-16835
SR-16835

Chemical Structure : SR-16835

CAS No.: 1207195-45-6

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SR-16835 (SR16835)

货号: PC-61540Not For Human Use, Lab Use Only.

SR-16835 is a potent full agonist of ORL1 receptor (NOP receptor) with binding Ki of 11.4 nM, with low-affinity mu-opioid partial agonist activity (Ki=79.9 nM).

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    SR-16835 is a potent full agonist of ORL1 receptor (NOP receptor) with binding Ki of 11.4 nM, with low-affinity mu-opioid partial agonist activity (Ki=79.9 nM).
    SR-16835 does not produce conditioned place preference (CPP) alone, but attenuates morphine CPP.
    SR-16835 shows antiallodynic activity in mice model of chronic pain.

    物理化学性质&存储条件

    分子量 386.54
    分子式 C26H30N2O
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    1-[1-(2,3,3a,4,5,6-Hexahydro-1H-phenalen-1-yl)-4-piperidinyl]-1,3-dihydro-2H-indol-2-one

    参考文献

    1. Toll L, et al. J Pharmacol Exp Ther. 2009 Dec;331(3):946-53.

    2. Khroyan TV, et al. J Pharmacol Exp Ther. 2011 Nov;339(2):687-93.

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