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首页-小分子抑制剂&激动剂-GPCR-Opioid Receptor-SR-16507
SR-16507

Chemical Structure : SR-16507

CAS No.: 1207195-44-5

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SR-16507 (SR16507)

货号: PC-61539Not For Human Use, Lab Use Only.

SR-16507 is a potent full agonist of ORL1 receptor (NOP receptor) and partial agonist of mu-opioid receptor with Ki of 5.22 nM and 1.07 nM, respectively.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    SR-16507 is a potent full agonist of ORL1 receptor (NOP receptor) and partial agonist of mu-opioid receptor with Ki of 5.22 nM and 1.07 nM, respectively.
    SR-16507  is a potent analgesic and produces conditioned place preference (CPP) alone, but also modestly attenuates morphine CPP; demonstrates antinociceptive effects in vivo.

    物理化学性质&存储条件

    分子量 368.565
    分子式 C24H36N2O
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    3-ethyl-1-(1-((1s,4s)-4-isopropylcyclohexyl)piperidin-4-yl)indolin-2-one

    参考文献

    1. Toll L, et al. J Pharmacol Exp Ther. 2009 Dec;331(3):946-53.

    2. Khroyan TV, et al. J Pharmacol Exp Ther. 2009 Dec;331(3):946-53.

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