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首页-小分子抑制剂&激动剂-Epigenetics-Bromodomain-SJ830599
SJ830599

Chemical Structure : SJ830599

CAS No.: 2215098-23-8

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SJ830599 (SJ 830599)

货号: PC-63255Not For Human Use, Lab Use Only.

SJ830599 is a modest selective BRD2-BD2 inhibitor with IC50 of 0.61 uM, 3.3-fold selectivity over BRD2-BD1.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    SJ830599 is a modest selective BRD2-BD2 inhibitor with IC50 of 0.61 uM, 3.3-fold selectivity over BRD2-BD1; demonstrates cytotoxicity against several pediatric cancer cell lines with EC50 values (HD-MB03 EC50=480 nM) comparable to BET inhibitor (BETi) clinical candidates.

    物理化学性质&存储条件

    分子量 356.422
    分子式 C20H24N2O4
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    Isopropyl ((2S,4R)-1-acetyl-6-(furan-2-yl)-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)carbamate

    参考文献

    1. Shadrick WR, et al. Bioorg Med Chem. 2018 Jan 1;26(1):25-36.

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