SGC2085 hydrochloride | PRMT4 (CARM1) inhibitor | Probechem Biochemicals

Chemical Structure : SGC2085 hydrochloride

CAS No.: 1821908-49-9

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SGC2085 hydrochloride (SGC-2085)

货号: PC-38535Not For Human Use, Lab Use Only.

SGC-2085 hydrochloride is a potent, selective protein arginine methyltransferase PRMT4 (CARM1) inhibitor with IC50 of 50 nM, displays >100-fold selectivity over other PRMTs (PRMT6 IC50=5.3 uM).

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1 mg	￥1580	In stock
5 mg	￥3280	In stock
10 mg	￥5280	In stock
25 mg		Get quote
100 mg		Get quote

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生物&药学活性

SGC-2085 hydrochloride is a potent, selective protein arginine methyltransferase PRMT4 (CARM1) inhibitor with IC50 of 50 nM, displays >100-fold selectivity over other PRMTs (PRMT6 IC50=5.3 uM).
SGC-2085 also shows complete selectivity against a panel of 21 human protein methyltransferases.

物理化学性质&存储条件

分子量	348.871
分子式	C19H25ClN2O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2S-amino-N-[[4-(3,5-dimethylphenoxy)-3-methylphenyl]methyl]-propanamide, monohydrochloride

参考文献

1. Ferreira de Freitas R, et al. J Med Chem. 2016 Jul 28;59(14):6838-47.

SGC2085 hydrochloride (SGC-2085)

生物&药学活性

物理化学性质&存储条件

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SGC2085 hydrochloride (SGC-2085)

生物&药学活性

物理化学性质&存储条件

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