SCH 58261 |CAS:160098-96-4 Probechem Biochemicals

Chemical Structure : SCH 58261

CAS No.: 160098-96-4

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SCH 58261 (SCH-58261;SCH58261)

货号: PC-45642Not For Human Use, Lab Use Only.

SCH 58261 is a potent and selective, competitive A2A adenosine receptor antagonist with Ki of 2.3 nM and 2.0 nM in rat and bovine brain, respectively.

规格	价格	库存
5 mg	￥780	In stock
10 mg	￥1180	In stock
25 mg	￥1980	In stock
50 mg	￥3480	In stock
100 mg		Get quote

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生物&药学活性

SCH 58261 is a potent and selective, competitive A2A adenosine receptor antagonist with Ki of 2.3 nM and 2.0 nM in rat and bovine brain, respectively.
SCH 58261 displays 323-, 53- and 100-fold selectivity over A1, A2B and A3 receptors, respectively.
SCH 58261 reverses reperfusion injury (IR) increased hippocampal Glu, GABA, glycine and aspartate, MPO, TNF-α, nitric oxide, and PGE in Male Wistar rats.

物理化学性质&存储条件

分子量	345.358
分子式	C18H15N7O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	DMSO: ≥ 34 mg/mL
Chemical Name/SMILES	7H-Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine, 2-(2-furanyl)-7-(2-phenylethyl)-

参考文献

1. Zocchi C, et al. J Pharmacol Exp Ther. 1996 Feb;276(2):398-404.

2. Beavis PA, et al. Proc Natl Acad Sci U S A. 2013 Sep 3;110(36):14711-6.

3. Mohamed RA, et al. Neurochem Res. 2012 Mar;37(3):538-47.

SCH 58261 (SCH-58261;SCH58261)

生物&药学活性

物理化学性质&存储条件

参考文献

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SCH 58261 (SCH-58261;SCH58261)

生物&药学活性

物理化学性质&存储条件

参考文献

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