SCH39166 |CAS:1227675-51-5 Probechem Biochemicals

Chemical Structure : SCH39166

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SCH39166 (SCH-39166;SCH 39166;Ecopipam)

货号: PC-60812Not For Human Use, Lab Use Only.

A potent, selective D1 dopamine receptor antagonist with Ki of 3.6 nM, >300-fold selectivity over D2 and 5-HT2 receptors.

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生物&药学活性

A potent, selective D1 dopamine receptor antagonist with Ki of 3.6 nM, >300-fold selectivity over D2 and 5-HT2 receptors; blocks dopamine-stimulated adenylate cyclase with Ki of 9.1 nM, inhibits both rat and squirrel monkey conditioned avoidance responding; antagonizes apomorphine-induced stereotypy in rats, demonstrates potential antipsychotic activity in vivo.

物理化学性质&存储条件

分子量	394.73
分子式	C19H20ClNO.HBr
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	6aS-trans)-11-Chloro-6,6a,7,8,9,13b-hexahydro-7-methyl-5H-benzo[d]naphth[2,1-b]azepin-12-ol hydrobromide

参考文献

1. Chipkin RE, et al. J Pharmacol Exp Ther. 1988 Dec;247(3):1093-102.

2. Lidow MS, et al. Brain Res. 1990 Dec 24;537(1-2):349-54.

3. Wu WL, et al. J Med Chem. 2005 Feb 10;48(3):680-93.

4. Criswell HE, et al. Neuropsychopharmacology. 1992 Sep;7(2):95-103.

SCH39166 (SCH-39166;SCH 39166;Ecopipam)

生物&药学活性

物理化学性质&存储条件

参考文献

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SCH39166 (SCH-39166;SCH 39166;Ecopipam)

生物&药学活性

物理化学性质&存储条件

参考文献

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