欢迎访问ProbeChem中文网站，英文网站请访问www.probechem.com
    英文 |     中文

产品咨询: sales@probechem.com
订购: order@probechem.com

首页-小分子抑制剂&激动剂-GPCR-Opioid Receptor-SCH221510
SCH221510

Chemical Structure : SCH221510

CAS No.: 322473-89-2

加入收藏

SCH221510 (SCH-221510)

货号: PC-60797Not For Human Use, Lab Use Only.

SCH221510 is a potent, selective, orally active nociceptin opioid receptor (NOP) agonist with EC50 of 12 nM, Ki of 0.3 nM.

规格 价格 库存 数量
10 mg Get quote
25 mg Get quote
50 mg Get quote
获取报价单
* 请选择数量再加入购物车
 or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    SCH221510 is a potent, selective, orally active nociceptin opioid receptor (NOP) agonist with EC50 of 12 nM, Ki of 0.3 nM.
    SCH221510 displays >50-fold over the mu-, kappa-, and delta-opioid receptors.
    SCH221510 produces anxiolytic-like effects in rats, does not disrupt overt behavior.

    物理化学性质&存储条件

    分子量 397.562
    分子式 C28H31NO
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    8-[bis(2-methylphenyl)-methyl]-3-phenyl-8-azabicyclo[3.2.1]octan-3-ol

    参考文献

    1. Varty GB, et al. J Pharmacol Exp Ther. 2008 Aug;326(2):672-82.

    2. Sobczak M, et al. J Pharmacol Exp Ther. 2014 Mar;348(3):401-9.

    3. Cremeans CM, et al. J Pharmacol Exp Ther. 2012 Oct;343(1):72-81.

    备案号：沪ICP备16042516号-1 Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

    联系我们 sales@probechem.com

    Bulk Inquiry

    * Indicates a Required FieldYour information is safe with us.

    • *Product name:
    • *Applicant name:
    • *Email address:
    • *Organization name:
    • *Requested quantity:
    • *Country:
    • *Additional Information:

    询单

    • *产品名称:
    • *姓名:
    • *邮箱:
    • *公司名称:
    • *询单数量:
    • *国籍:
    • 询单信息: