SB 206553 | 5-HT2B/5-HT2C antagonist | Probechem Biochemicals

Chemical Structure : SB 206553

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SB 206553 (SB206553)

货号: PC-62760Not For Human Use, Lab Use Only.

SB 206553 is a potent and selective 5-HT2B/5-HT2C receptor antagonist with pA2 of 8.89 for rat 5-HT2B, pKi of 7.92 for human 5-HT2C, displays >80-fold selectivity over other 5-HT receptor subtypes.

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生物&药学活性

SB 206553 is a potent and selective 5-HT2B/5-HT2C receptor antagonist with pA2 of 8.89 for rat 5-HT2B, pKi of 7.92 for human 5-HT2C, displays >80-fold selectivity over other 5-HT receptor subtypes.
SB 206553 exhibits anxiolytic-like properties both in vitro and in vivo.

物理化学性质&存储条件

分子量	328.80
分子式	C17H17ClN4O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3,5-Dihydro-5-methyl-N-3-pyridinylbenzo[1,2-b:4,5-b']dipyrrole-1(2H)-carboxamide hydrochloride

参考文献

1. Forbes IT, et al. J Med Chem. 1995 Jul 7;38(14):2524-30.

2. Upton N, et al. Eur J Pharmacol. 1998 Oct 16;359(1):33-40.

3. Kennett GA, et al. Br J Pharmacol. 1996 Feb;117(3):427-434.

4. Porras G, et al. Neuropsychopharmacology. 2002 Mar;26(3):311-24.

SB 206553 (SB206553)

生物&药学活性

物理化学性质&存储条件

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SB 206553 (SB206553)

生物&药学活性

物理化学性质&存储条件

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