SB-277011 hydrochloride | D3R antagonist | Probechem Biochemicals

Chemical Structure : SB-277011 hydrochloride

CAS No.: 215804-67-4

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SB-277011 hydrochloride (SB277011A hydrochloride)

货号: PC-23120Not For Human Use, Lab Use Only.

SB-277011 hydrochloride (SB277011A) is a potent and selective dopamine D3 receptor antagonist with pKi of 8.0.

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10 mg	￥1280	In stock
25 mg	￥2180	In stock
50 mg	￥3680	In stock
100 mg		Get quote

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生物&药学活性

SB-277011 hydrochloride (SB277011A) is a potent and selective dopamine D3 receptor antagonist with pKi of 8.0.
SB-277011 displays >100-fold selectivity against the D2, 5-HT1B, and 5-HT1D receptors.
SB-277011 exhibits high oral bioavailability and brain penetration in rats.

物理化学性质&存储条件

分子量	475.03
分子式	C28H31ClN4O
外观性状	Solid
CAS No.
储存条件	固体粉末 -20°C 12 个月; 4°C 6 个月	配置液 -80°C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-((1r,4r)-4-(2-(6-cyano-3,4-dihydroisoquinolin-2(1H)-yl)ethyl)cyclohexyl)quinoline-4-carboxamide hydrochloride

参考文献

1. Stemp G, et al. J Med Chem. 2000 May 4;43(9):1878-85.

2. Reavill C, et al. J Pharmacol Exp Ther. 2000 Sep;294(3):1154-65.

3. Ashby CR Jr, et al. J Pharmacol Exp Ther. 2000 Sep;294(3):1166-74.

SB-277011 hydrochloride (SB277011A hydrochloride)

生物&药学活性

物理化学性质&存储条件

参考文献

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SB-277011 hydrochloride (SB277011A hydrochloride)

生物&药学活性

物理化学性质&存储条件

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