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首页-小分子抑制剂&激动剂-Others-Other Targets-SAN9812
SAN9812

Chemical Structure : SAN9812

CAS No.:

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SAN9812 (SAN-9812;Carnostatine)

货号: PC-35233Not For Human Use, Lab Use Only.

SAN9812 (Carnostatine) is a potent, highly selective, competitive inhibitor of Carnosinase 1 (CN1) activity with Ki of 11 nM.

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25 mg ￥5850 In stock
100 mg ￥12800 In stock
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

SAN9812 (Carnostatine) is a potent, highly selective, competitive inhibitor of Carnosinase 1 (CN1) activity with Ki of 11 nM; displays no activity against a standard panel of 33 different receptors, channels, transporters and enzymes; inhibits human recombinant CN1 at a carnosine concentration of 200 µM with IC50 of 18 nM, also demonstrates inhibitory activity on human CN1 in serum from TG mice-expressing human CN1 and serum from healthy human volunteers with IC50 of 650 and 340 nM, respectively; increases carnosine levels in plasma and kidney in mice.

物理化学性质&存储条件

分子量 256.262
分子式 C10H16N4O4
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

((S)-4-amino-2-hydroxybutanoyl)-L-histidine

参考文献

1. Qiu J, et al. Amino Acids. 2018 Jun 20. doi: 10.1007/s00726-018-2601-z.

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