S-17092 |CAS:176797-26-5 Probechem Biochemicals

Chemical Structure : S-17092

加入收藏

S-17092 (S17092;S 17092)

货号: PC-70065Not For Human Use, Lab Use Only.

A highly potent, specific and cell permeant inhibitor of human proline endopeptidase (PE) with Ki of 1 nM.

规格	价格	库存	数量
25 mg		Get quote
100 mg		Get quote
500 mg		Get quote
1 g		Get quote

获取报价单

* 请选择数量再加入购物车

or Bulk Inquiry

大包装，大折扣！

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

生物&药学活性

A highly potent, specific and cell permeant inhibitor of human proline endopeptidase (PE) with Ki of 1 nM; shows no activity against a series of other peptidases including aminopeptidases B and M, dipeptidylaminopeptidase IV, endopeptidases, calpains and angiotensin-converting enzyme; significantly increases in SP- and alpha-MSH-like immunoreactivity in the frontal cortex and hypothalamus in rats (30mg/kg); shows cognition-enhancing properties in chronic low dose MPTP-treated monkeys.

物理化学性质&存储条件

分子量	384.53
分子式	C22H28N2O2S
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	((2S,3aS,7aS)-1-((1R,2R)-2-phenylcyclopropane-1-carbonyl)octahydro-1H-indol-2-yl)(thiazolidin-3-yl)methanone

参考文献

1. Barelli H, et al. Biochem Biophys Res Commun. 1999 Apr 21;257(3):657-61.

2. Bellemère G, et al. J Neurochem. 2003 Mar;84(5):919-29.

3. Schneider JS, et al. Neuropsychopharmacology. 2002 Feb;26(2):176-82.

S-17092 (S17092;S 17092)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

S-17092 (S17092;S 17092)

生物&药学活性

物理化学性质&存储条件

参考文献

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

询单

Get Quotation Now

* Indicates a Required FieldYour information is safe with us.