Ralaniten acetate | AR-NTD inhibitor | Probechem Biochemicals

Chemical Structure : Ralaniten acetate

CAS No.: 1637573-04-6

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Ralaniten acetate (EPI-506, EPI 506, EPI506)

货号: PC-60530Not For Human Use, Lab Use Only.

Ralaniten acetate (EPI-506) is the acetate prodrug of Ralaniten (EPI-002), a small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor for the treatment of advanced prostate cancer.

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10 mg	￥5880	In stock
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生物&药学活性

Ralaniten acetate (EPI-506) is the acetate prodrug of Ralaniten (EPI-002), a small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor for the treatment of advanced prostate cancer.
AR NTD-targeting agents have the potential to overcome shortcomings of current hormonal therapies by inhibiting all forms of AR-mediated transcriptional activity, and as a result, may affect a broader AR population including mutational and splice variant ARs.

物理化学性质&存储条件

分子量	521.003
分子式	C27H33ClO8
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-3-(4-(2-(4-((S)-2-acetoxy-3-chloropropoxy)phenyl)propan-2-yl)phenoxy)propane-1,2-diyl diacetate

参考文献

1. Antonarakis ES, et al. Oncologist. 2016 Dec;21(12):1427-1435.

Ralaniten acetate (EPI-506, EPI 506, EPI506)

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物理化学性质&存储条件

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Ralaniten acetate (EPI-506, EPI 506, EPI506)

生物&药学活性

物理化学性质&存储条件

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