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首页-小分子抑制剂&激动剂-Nuclear Receptor/Transcription Factor-Androgen Receptor (AR)-Ralaniten
Ralaniten

Chemical Structure : Ralaniten

CAS No.: 1203490-23-6

Ralaniten (EPI-002)

货号: PC-60529Not For Human Use, Lab Use Only.

Ralaniten (EPI-002) is a novel small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor, inhibits AR transcriptional activity with IC50 of 7.4 uM.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

Ralaniten (EPI-002) is a novel small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor, inhibits AR transcriptional activity with IC50 of 7.4 uM.
AR NTD-targeting agents have the potential to overcome shortcomings of current hormonal therapies by inhibiting all forms of AR-mediated transcriptional activity, and as a result, may affect a broader AR population including mutational and splice variant ARs.

物理化学性质&存储条件

分子量 394.89
分子式 C21H27ClO5
外观性状 Solid
CAS No.
储存条件
固体粉末
-20 °C 12 个月; 4°C 6 个月
配置液
-80 °C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

(2R)-3-[4-(2-{4-[(2S)-3-chloro- 2-hydroxypropoxy]phenyl}propan-2-yl)phenoxy]propane- 1,2-diol

参考文献

1. Antonarakis ES, et al. Oncologist. 2016 Dec;21(12):1427-1435.

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