Chemical Structure : Ralaniten
CAS No.: 1203490-23-6
货号: PC-60529Not For Human Use, Lab Use Only.
Ralaniten (EPI-002) is a novel small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor, inhibits AR transcriptional activity with IC50 of 7.4 uM.
规格 | 价格 | 库存 | 数量 |
---|---|---|---|
5 mg | ¥880 | In stock | |
10 mg | ¥1280 | In stock | |
25 mg | ¥2180 | In stock | |
50 mg | ¥3580 | In stock | |
100 mg | Get quote |
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Ralaniten (EPI-002) is a novel small-molecule inhibitor of androgen receptor (AR) N-terminal domain inhibitor, inhibits AR transcriptional activity with IC50 of 7.4 uM.
AR NTD-targeting agents have the potential to overcome shortcomings of current hormonal therapies by inhibiting all forms of AR-mediated transcriptional activity, and as a result, may affect a broader AR population including mutational and splice variant ARs.
分子量 | 394.89 | |
分子式 | C21H27ClO5 | |
外观性状 | Solid | |
储存条件 |
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|
Solubility |
10 mM in DMSO |
|
Chemical Name/SMILES |
(2R)-3-[4-(2-{4-[(2S)-3-chloro- 2-hydroxypropoxy]phenyl}propan-2-yl)phenoxy]propane- 1,2-diol |
1. Antonarakis ES, et al. Oncologist. 2016 Dec;21(12):1427-1435.
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