RY796 racemate |CAS:854165-96-1 Probechem Biochemicals

Chemical Structure : RY796 racemate

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RY796 racemate (RY 796;RY-796)

货号: PC-60805Not For Human Use, Lab Use Only.

A novel potent, selective Kv2 channel inhibitor that potently inhibits Kv2.1 and Kv2.2 with IC50 of 0.14 and 0.09 uM, respectively.

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生物&药学活性

A novel potent, selective Kv2 channel inhibitor that potently inhibits Kv2.1 and Kv2.2 with IC50 of 0.14 and 0.09 uM, respectively; shows no significant activity against Kv1.2 and Kv7.1, and Cav channels; enhances GSIS in isolated wild-type (WT) mouse and human islets, but not in islets from Kv2.1(-/-) mice, enhances somatostatin release in isolated human and mouse islets.

物理化学性质&存储条件

分子量	353.466
分子式	C21H27N3O2
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-(dimethylamino)-5-isobutyramido-N-(1-phenylethyl)benzamide

参考文献

1. Herrington J, et al. Mol Pharmacol. 2011 Dec;80(6):959-64.

2. Li XN, et al. J Pharmacol Exp Ther. 2013 Feb;344(2):407-16.

RY796 racemate (RY 796;RY-796)

生物&药学活性

物理化学性质&存储条件

参考文献

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RY796 racemate (RY 796;RY-796)

生物&药学活性

物理化学性质&存储条件

参考文献

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