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首页-小分子抑制剂&激动剂-GPCR-Orexin Receptor-RTOXA-43
RTOXA-43

Chemical Structure : RTOXA-43

CAS No.: 2832067-72-6

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RTOXA-43 (RTOXA43)

货号: PC-20563Not For Human Use, Lab Use Only.

RTOXA-43 is a potent, dual orexin receptor agonist with EC50 of 24 nM at both OX2R and OX1R.

规格 价格 库存 数量
2 mg ￥2180 In stock
5 mg ￥3780 In stock
10 mg ￥5880 In stock
25 mg Get quote
50 mg Get quote
100 mg Get quote
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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

生物&药学活性

RTOXA-43 is a potent, dual orexin receptor agonist with EC50 of 24 nM at both OX2R and OX1R.
RTOXA-43 (40 mg/kg, i.p.) increased time awake, decreased time asleep and increased sleep/wake consolidation when measured using continuous EEG/EMG recordings in 12-month old mice.

物理化学性质&存储条件

分子量 663.79
分子式 C37H37N5O5S
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

4'-methoxy-N-methyl-3'-(N-(3-((2-(3-methylbenzamido)ethyl)amino)phenyl)sulfamoyl)-N-(pyridin-4-ylmethyl)-[1,1'-biphenyl]-3-carboxamide

参考文献

1. Dehui Zhang, et al. J Med Chem. 2021 Jun 24;64(12):8806-8825.

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