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首页-小分子抑制剂&激动剂-Others-Other Targets-RTI-263
RTI-263

Chemical Structure : RTI-263

CAS No.:

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RTI-263 (SerPheLysAsn-NH2)

货号: PC-21471Not For Human Use, Lab Use Only.

RTI-263 (SerPheLysAsn-NH2) is a potent, selective tetrapeptide neuropeptide S receptor (NPSR, GPR154) biased agonist with EC50 of 3.02 nM for hNPSR calcium mobilization.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

RTI-263 (SerPheLysAsn-NH2) is a potent, selective tetrapeptide neuropeptide S receptor (NPSR, GPR154) biased agonist with EC50 of 3.02 nM for hNPSR calcium mobilization.
RTI-263 greatly attenuated hyperlocomotor stimulation in vivo but retains activity in assays that correlate with memory consolidation and anxiolytic activity.
RTI-263 has a bias for the calcium mobilization pathway, at the human and mouse NPSR receptor.

物理化学性质&存储条件

分子量 493.57
分子式 C22H35N7O6
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

(S)-2-((S)-6-amino-2-((S)-2-((S)-2-amino-3-hydroxypropanamido)-3-phenylpropanamido)hexanamido)succinamide

参考文献

1. Stewart D Clark, et al. Neuropharmacology. 2017 May 15:118:69-78.

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