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首页-小分子抑制剂&激动剂-GPCR-Opioid Receptor-R995045
R995045

Chemical Structure : R995045

CAS No.: 1285536-79-9

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R995045 (R 995045, R-995045)

货号: PC-72734Not For Human Use, Lab Use Only.

R995045 is a novel δ-opioid receptor (δOR) agonist with pKi of 5.94, cAMP pIC50 of 6.01, >10-fold selectivity over µOR and κOR.

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纯度 & COA & 质检文件 纯度: >98% (HPLC)

生物&药学活性

R995045 is a novel δ-opioid receptor (δOR) agonist with pKi of 5.94, cAMP pIC50 of 6.01, >10-fold selectivity over µOR and κOR.
R995045 acts as a negative allosteric modulator for leu-enkephalin potency in the cAMP glosensor assay.

物理化学性质&存储条件

分子量 342.373
分子式 C16H14N4O3S
外观性状 Solid
CAS No.
储存条件
固体粉末
-20°C 12 个月; 4°C 6 个月
配置液
-80°C 6 个月; -20°C 6 个月
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

N'-(2-hydroxy-3-methoxybenzylidene)-3-(2-thienyl)-1H-pyrazole-5-carbohydrazide

参考文献

1. Meqbil YJ, et al. Molecules. 2021 Nov 29;26(23):7236.

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