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首页-小分子抑制剂&激动剂-Tyrosine Kinase-TAM Receptor (Tyro3-Axl-Mer)-R916562
R916562

Chemical Structure : R916562

CAS No.: 1037798-41-6

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R916562 (R 916562;R-916562;R562)

货号: PC-35348Not For Human Use, Lab Use Only.

R916562 (R562) is a potent, dual Axl/VEGFR2 inhibitor with celluar IC50 of 136 nM for Axl.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    R916562 (R562) is a potent, dual Axl/VEGFR2 inhibitor with celluar IC50 of 136 nM for Axl.
    R916562 blocks growth of MDA-MB-231 breast carcinomas implanted subcutaneously in nu/nu mice.
    R916562 also shows efficacy in the Caki-1 human renal carcinoma xenograft model.

    物理化学性质&存储条件

    分子量 536.099
    分子式 C26H30ClN9S
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    1H-1,2,4-Triazole-3,5-diamine, N3-[4-[4-(1R,2R,4S)-bicyclo[2.2.1]hept-2-yl-1-piperazinyl]phenyl]-1-(2-chloro-7-methylthieno[3,2-d]pyrimidin-4-yl)-

    参考文献

    1. Goff D, et al. Bioorg Med Chem Lett. 2017 Aug 15;27(16):3766-3771.

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