R-283 (R283, TG2-IN-1)

Chemical Structure : R-283

CAS No.: 135273-74-4

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货号: PC-61734Not For Human Use, Lab Use Only.

R-283 is a potent and selective human tissue transglutaminase (hTG2) inhibitor with IC50 of 4 uM..

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R-283 (R283, TG2-IN-1) is a potent and selective human tissue transglutaminase (hTG2) inhibitor with IC50 of 4 uM.

分子量	220.715
分子式	C8H13ClN2OS
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1,3-dimethyl-2-((2-oxopropyl)thio)-1H-imidazol-3-ium chloride

1. Griffin M, et al. Bioorg Med Chem Lett. 2008 Oct 15;18(20):5559-62.

2. Freund KF, et al. Biochemistry. 1994 Aug 23;33(33):10109-19.

3. Miura A, et al. J Biol Chem. 2013 Nov 8;288(45):32720-30.