QCA276 |CAS:2126819-40-5 Probechem Biochemicals

Chemical Structure : QCA276

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QCA276 (QCA 276;QCA-276)

货号: PC-35400Not For Human Use, Lab Use Only.

QCA276 is a novel potent BET proteins inhibitor with IC50/Ki of 10/.3 nM, QCA276 is the BET ligand for PROTAC QCA570.

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生物&药学活性

QCA276 is a novel potent BET proteins inhibitor with IC50/Ki of 10/.3 nM, QCA276 is the BET ligand for PROTAC QCA570; effectively inhibits human BRD2, BRD3, and BRD4 BD1 and BD2 proteins with Ki of 2-20 nM.

物理化学性质&存储条件

分子量	401.488
分子式	C22H19N5OS
外观性状	Solid
CAS No.
储存条件	固体粉末 -20 °C 12 个月; 4°C 6 个月	配置液 -80 °C 6 个月; -20°C 6 个月
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	3-Benzyl-9-methyl-2-((1-methyl-1H-pyrazol-4-yl)ethynyl)-4H,6Hthieno[2,3-e][1,2,4]triazolo[3,4-c][1,4]oxazepine

参考文献

1. Qin C, et al. J Med Chem. 2018 Jul 18. doi: 10.1021/acs.jmedchem.8b00506.

QCA276 (QCA 276;QCA-276)

生物&药学活性

物理化学性质&存储条件

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QCA276 (QCA 276;QCA-276)

生物&药学活性

物理化学性质&存储条件

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