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首页-小分子抑制剂&激动剂-Metabolic Enzyme/Protease-Phosphodiesterase (PDE)-PyP-1
PyP-1

Chemical Structure : PyP-1

CAS No.: 1370527-16-4

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PyP-1 (PyP1)

货号: PC-62700Not For Human Use, Lab Use Only.

PyP-1 is a potent, highly selective, and orally bioavailable PDE10A inhibitor with Ki of 0.23 nM.

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纯度 & COA & 质检文件 纯度: >98% (HPLC) Select Batch:

    生物&药学活性

    PyP-1 is a potent, highly selective, and orally bioavailable PDE10A inhibitor with Ki of 0.23 nM.
    PyP-1 exhibits excellent pharmacokinetic and physicochemical properties, and a clean off-target profile.
    PyP-1 displays in vivo preclinical target engagement and clean preclinical profile

    物理化学性质&存储条件

    分子量 375.436
    分子式 C20H21N7O
    外观性状 Solid
    CAS No.
    储存条件
    固体粉末
    -20 °C 12 个月; 4°C 6 个月
    配置液
    -80 °C 6 个月; -20°C 6 个月
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    N-((1-methyl-1H-pyrazol-4-yl)methyl)-5-(((1S,2S)-2-(pyridin-2-yl)cyclopropyl)methoxy)pyrazolo[1,5-a]pyrimidin-7-amine

    参考文献

    1. Raheem IT, et al. Bioorg Med Chem Lett. 2016 Jan 1;26(1):126-32.

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